A Menin-MLL Inhibitor Induces Specific Chromatin Changes and Eradicates Disease in Models of MLL-Rearranged Leukemia - ScienceDirect

Inhibition of the Menin (MEN1) and MLL (MLL1, KMT2A) interaction is a potential therapeutic strategy for MLL-rearranged (MLL-r) leukemia. Structure-ba…

Menin-MLL inhibitors reverse oncogenic activity of MLL fusion

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MLL::AF9 degradation induces rapid changes in transcriptional

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Recent Progress of Small Molecule Menin–MLL Interaction Inhibitors

A novel Menin-MLL1 inhibitor, DS-1594a, prevents the progression

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The menin-MLL1 interaction is a molecular dependency in NUP98

A Menin-MLL Inhibitor Induces Specific Chromatin Changes and

Pharmacologic Inhibition of the Menin-MLL Interaction Blocks